SCHEMBL27596191

SCHEMBL27596191

O=C(OCCCNc1ncc(C(=O)c2ccccc2C(F)(F)F)s1)c1cccs1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
CTNNB1 P35222 1/20 0.42
WNT3A P56704 1/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
GLA P06280 1/20 0.38
BRCA1 P38398 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27596182 0.90 MAPK13 (0.43) CTNNB1WNT3AALDH1A1LMNAGLA
SCHEMBL27596328 0.88 MAPK13 (0.51) ALDH1A1MAPT
SCHEMBL27596193 0.88 PKM (0.44) CTNNB1WNT3AALDH1A1LMNASMN1; SMN2
SCHEMBL27596183 0.87 ALDH1A1 (0.40) HTTALDH1A1LMNAKDM4EMAPT
SCHEMBL27615061 0.82 LIMK1 (0.41)
SCHEMBL27596189 0.81 MAPK13 (0.37)
SCHEMBL5564938 0.81 MAPK13 (0.44)
SCHEMBL27614965 0.79 ALDH1A1 (0.44) ALDH1A1LMNASMN1; SMN2KDM4EMAPT
SCHEMBL27596159 0.78 MAPK13 (0.44)
SCHEMBL5564934 0.77 MAPK13 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN disclosed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN disclosed