SCHEMBL27596193

SCHEMBL27596193

Cc1ccccc1C(=O)c1cnc(NCCCOC(=O)c2cccs2)s1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.44
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
LCK P06239 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
THRB P10828 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MAPK14 Q16539 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27596183 0.90 ALDH1A1 (0.40) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL27596328 0.89 MAPK13 (0.51) ALDH1A1MAPTMAPK14
SCHEMBL27596182 0.89 MAPK13 (0.43) CTNNB1WNT3AALDH1A1LMNANPC1
SCHEMBL27596191 0.88 HTT (0.44) CTNNB1WNT3AALDH1A1MAPTMEN1
SCHEMBL27614965 0.88 ALDH1A1 (0.44) LCKALDH1A1MAPTMEN1KMT2A
SCHEMBL27614917 0.82 F2 (0.37) ALDH1A1KDM4EMAPK14
SCHEMBL27596205 0.82 MAPK14 (0.43) LCKMAPK14
SCHEMBL27614981 0.80 MAPK14 (0.41) NPC1RAB9AMAPK14
SCHEMBL27615012 0.79 MAPK14 (0.42) MAPK14
SCHEMBL5563877 0.79 NPC1 (0.46) LCKMAPTNPC1RAB9AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN disclosed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN disclosed