SCHEMBL27596453

SCHEMBL27596453

[CH2]CC1CCN(Cc2ccccc2)CC1=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.49
CCR3 P51677 1/20 0.47
SIGMAR1 Q99720 2/20 0.46
HTR2A P28223 1/20 0.46
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
HTR1A P08908 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5975118 0.86 CCR3 (0.57) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL5974931 0.86 CCR3 (0.57) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL5974936 0.86 CCR3 (0.57) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL31288163 0.85 ACHE (0.53) ACHECCR3SIGMAR1HTR2ADRD2
Hydrochloric Acid SCHEMBL6660125 0.85 CCR3 (0.55) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL3572183 0.82 MEN1 (0.48) ACHECCR3SIGMAR1DRD2DRD4
SCHEMBL11178158 0.81 DRD2 (0.49) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL995393 0.80 ACHE (0.50) ACHESIGMAR1
SCHEMBL5974372 0.79 LMNA (0.55) ACHECCR3SIGMAR1HTR2ADRD2
SCHEMBL5974378 0.79 LMNA (0.55) ACHECCR3SIGMAR1HTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699008-A Sulfamide derivative and pharmaceutical composition containing it EA制药株式会社 2018-10-23 CN disclosed
CN-104540826-B Spiro-fused piperidine derivatives useful as inhibitors of extrarenal potassium channels 默沙东公司 2018-04-20 CN disclosed
CN-107459508-A Annelated pyrimidines as the inhibitor of P97 compounds 克里弗生物科学公司 2017-12-12 CN disclosed
CN-101434596-A Novel azaheterocyclic amides useful for treating pain ABBOTT LAB (US) 2009-05-20 CN disclosed
CN-1849315-A Novel nitrogen-containing heterocyclic amides for the treatment of pain ABBOTT LAB (US) 2006-10-18 CN disclosed
CN-1826334-A Tetrahydropyranyl cyclopentyl heterocyclic amide modulators of chemokine receptor activity MERCK & CO INC (US) 2006-08-30 CN disclosed
CN-1481377-A Cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteinases and TNF-alpha ����˹�ж�-����˹˹����ҩƷ��˾ 2004-03-10 CN disclosed