SCHEMBL27599208

SCHEMBL27599208

COc1ccc2c(c1)c(CC(=O)OOC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](C=O)NC(C)=O)c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.62
AKR1C3 P42330 2/20 0.62
CNR2 P34972 1/20 0.62
PTGS1 P23219 2/20 0.56
KDM4E B2RXH2 1/20 0.56
MEN1 O00255 1/20 0.56
PTGES O14684 1/20 0.56
ABCC3 O15438 1/20 0.56
ABCC4 O15439 1/20 0.56
ABCB11 O95342 1/20 0.56
MT-CO2 P00403 1/20 0.56
LMNA P02545 1/20 0.56
ALB P02768 1/20 0.56
CYP1A2 P05177 1/20 0.56
ABCB1 P08183 1/20 0.56
ALOX5 P09917 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
CXCL8 P10145 1/20 0.56
AR P10275 1/20 0.56
CYP2D6 P10635 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glucametacin SCHEMBL30344903 0.86 PTGS2 (0.72) PTGS2
Glucametacin SCHEMBL27641193 0.86 PTGS2 (0.72) PTGS2
Glucametacin SCHEMBL5081097 0.86 PTGS2 (0.72) PTGS2
Glucametacin SCHEMBL24511 0.86 PTGS2 (0.72) PTGS2
SCHEMBL11263049 0.79 PTGS2 (0.74) PTGS2AKR1C3CNR2PTGS1KDM4E
SCHEMBL27617617 0.79 PTGS2 (0.65) PTGS2AKR1C3CNR2PTGS1GLO1
SCHEMBL14086813 0.78 PTGS2 (1.00) PTGS2AKR1C3CNR2PTGS1KDM4E
SCHEMBL30426824 0.78 PTGS2 (1.00) PTGS2AKR1C3CNR2PTGS1KDM4E
Glucametacin SCHEMBL9988209 0.78 PTGS2 (0.63) PTGS2
Indomethacin SCHEMBL8509782 0.77 PTGS2 (0.74) PTGS2AKR1C3CNR2PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1616474-A Acetamido glucose devicative of indomethacin and its synthetic method and use CHINA OCEANOGRAPHIC UNIV (CN) 2005-05-18 CN disclosed