SCHEMBL27600987

SCHEMBL27600987

COC(=O)c1ccc(CCBr)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CCR6 P51684 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
CYP4F2 P78329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6618508 0.88 ALDH1A1 (0.46) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL489064 0.87 ALDH1A1 (0.45) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL4451323 0.86 TSHR (0.47) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL7219535 0.86 NPC1 (0.44) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL3921415 0.86 CYP4A11 (0.54) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL27523349 0.85 GAA (0.50) FFAR4ALDH1A1GAAKDM4EMAPT
Hydrochloric Acid SCHEMBL12499751 0.84 LMNA (0.47) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL8252765 0.83 GAA (0.47) FFAR4ALDH1A1GAAKDM4EMAPT
SCHEMBL23582779 0.83 FFAR4 (0.61) FFAR4ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL18030873 0.83 PLA2G2A (0.53) FFAR4ALDH1A1GAAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101896470-B Dual-acting benzimidazole derivatives and their use as antihypertensive agents THERAVANCE INC 2013-04-10 CN disclosed
CN-101896470-A Dual-acting benzimidazole derivatives and their use as antihypertensive agents THERAVANCE INC 2010-11-24 CN disclosed
CN-1922151-A Substituted azole derivatives, compositions, and methods of use TRANSTECH PHARMA INC (US) 2007-02-28 CN disclosed
CN-1606553-A Oxytocin agonistenoxytocin agonisten FERRING BV (NL) 2005-04-13 CN disclosed