SCHEMBL27608342

SCHEMBL27608342

Cc1c(N)cccc1OC(=O)NC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.39
PIK3CA P42336 1/20 0.39
HTR1A P08908 2/20 0.39
DRD2 P14416 2/20 0.39
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 3/20 0.36
PGR P06401 1/20 0.36
GAA P10253 1/20 0.36
PTGS1 P23219 1/20 0.36
MAPK1 P28482 1/20 0.36
ESR1 P03372 1/20 0.35
KCNH2 Q12809 1/20 0.35
KDM4E B2RXH2 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CFTR P13569 1/20 0.34
POLB P06746 2/20 0.34
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL248601 0.85 SMN1; SMN2 (0.44) ACHETSHRHTR1ADRD2ALDH1A1
SCHEMBL29286690 0.83 HTR1A (0.36) ACHEHTR1ADRD2ALDH1A1HSD17B10
SCHEMBL27698905 0.81 MAPK1 (0.44) CYP3A4HTR1ADRD2ALDH1A1PGR
SCHEMBL27611466 0.81 HTR1A (0.39) HTR1ADRD2ALDH1A1HSD17B10PGR
SCHEMBL907658 0.78 ACHE (0.61) ACHETSHRCYP3A4PIK3CAALDH1A1
SCHEMBL23420829 0.78 TDP1 (0.50) TSHRALDH1A1GAAMAPK1KDM4E
SCHEMBL25295423 0.77 ATM (0.42) ACHEALDH1A1HSD17B10PGRGAA
SCHEMBL27767915 0.75 ALDH1A1 (0.47) CYP3A4ALDH1A1HSD17B10SMN1; SMN2LMNA
SCHEMBL29131348 0.75 MAPK1 (0.41) HTR1ADRD2ALDH1A1HSD17B10PGR
SCHEMBL11485248 0.75 KMT2A (0.50) ALDH1A1HSD17B10KDM4ESMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101460508-A Thiazolyl-dihydro-chinazoline BOEHRINGER INGELHEIM INT (DE) 2009-06-17 CN disclosed
CN-1568187-A 2H-2,3-dinitrogen phenodiazine-1-ketone and using method thereof ICOS CORP (US) 2005-01-19 CN disclosed