SCHEMBL27612752

SCHEMBL27612752

NC(=O)Cc1cccnc1CC(N)=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 1/20 0.44
MAPT P10636 1/20 0.44
GAA P10253 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 4/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTK2 Q05397 4/20 0.38
PARP1 P09874 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTT P42858 1/20 0.37
NAPRT Q6XQN6 1/20 0.36
P2RX7 Q99572 2/20 0.36
ITK Q08881 1/20 0.36
CA2 P00918 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542523 0.87 KDM4E (0.41) KDM4ECYP1A2MAPTGAANPSR1
SCHEMBL29394811 0.83 PAX8 (0.43) KDM4ECYP1A2MAPTL3MBTL1HTT
SCHEMBL4668812 0.81 L3MBTL1 (0.57) KDM4ECYP1A2MAPTGAANPSR1
SCHEMBL1515657 0.81 KDM4E (0.44) KDM4ECYP1A2MAPTGAANPSR1
SCHEMBL25243173 0.79 MAPT (0.42) KDM4ECYP1A2MAPTALDH1A1L3MBTL1
SCHEMBL2334108 0.79 ALDH1A1 (0.38) KDM4ECYP1A2MAPTALDH1A1L3MBTL1
SCHEMBL2178576 0.79 SMN1; SMN2 (0.47) KDM4ECYP1A2MAPTALDH1A1L3MBTL1
SCHEMBL31439135 0.79 PARP1 (0.51) KDM4EMAPTNPSR1ALDH1A1L3MBTL1
SCHEMBL999250 0.79 P2RX7 (0.50) KDM4ECYP1A2MAPTALDH1A1PARP1
SCHEMBL6513742 0.79 PLAU (0.44) MAPTL3MBTL1HTTP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1678321-A Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds RIGEL PHARMACEUTICALS INC (US) 2005-10-05 CN disclosed