SCHEMBL27615288

SCHEMBL27615288

C#Cc1cc([N+](=O)[O-])ccc1C(=O)OC(=O)C(=C)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
NR1H4 Q96RI1 2/20 0.37
ADRB2 P07550 2/20 0.36
ADRB1 P08588 2/20 0.36
ADRB3 P13945 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 4/20 0.35
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 3/20 0.34
HPGD P15428 2/20 0.34
VCAM1 P19320 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27552998 0.84 ALDH1A1 (0.41) ALDH1A1TDP1CYP3A4ALOX15NR1H4
SCHEMBL27462168 0.82 ADRB2 (0.52) ALDH1A1TDP1CYP3A4ALOX15NR1H4
SCHEMBL4036027 0.82 ALDH1A1 (0.42) ALDH1A1TDP1CYP3A4ALOX15NR1H4
SCHEMBL27615290 0.81 NR1H4 (0.55) ALDH1A1TDP1NR1H4ADRB2ADRB1
SCHEMBL27615400 0.81 NR1H4 (0.39) ALDH1A1TDP1CYP3A4ALOX15NR1H4
SCHEMBL27615287 0.79 CES2 (0.36) ALDH1A1TDP1CYP3A4ALOX15NR1H4
SCHEMBL27563637 0.79 GAA (0.52) ALDH1A1CYP3A4ALOX15NR1H4SMN1; SMN2
SCHEMBL27487269 0.74 POLB (0.50) ALDH1A1TDP1NR1H4ADRB2ADRB1
SCHEMBL4030328 0.74 ALDH1A1 (0.58) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2
SCHEMBL27449894 0.73 ALDH1A1 (0.55) ALDH1A1TDP1CYP3A4ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343238-C Quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1585754-A Quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2005-02-23 CN disclosed