SCHEMBL27623744

SCHEMBL27623744

CC(=O)Oc1cc2c(Br)nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c2cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.36
MAPK1 P28482 2/20 0.36
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 3/20 0.33
HSD17B10 Q99714 3/20 0.33
HPGD P15428 2/20 0.33
USP2 O75604 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 3/20 0.33
ESR1 P03372 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
HMGB1 P09429 1/20 0.33
GGT1 P19440 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27623653 0.84 BACE1 (0.34) BACE1MAPK1CYP4F2CYP4A11KDM4E
SCHEMBL4149112 0.80 MAPK1 (0.39) MAPK1KDM4EALDH1A1USP2SMN1; SMN2
SCHEMBL27604769 0.79 BACE1 (0.34) BACE1MAPK1KDM4EALDH1A1HSD17B10
SCHEMBL27604940 0.77 NTSR1 (0.35) MAPK1KDM4EALDH1A1NPC1RAB9A
SCHEMBL4139741 0.74 VCAM1 (0.34) KDM4EALDH1A1SMN1; SMN2BLMTDP1
SCHEMBL16620077 0.73 ALDH1A1 (0.37) MAPK1KDM4EALDH1A1CYP2C19MAPT
SCHEMBL1199662 0.73 MAPK1 (0.36) MAPK1KDM4EALDH1A1CYP2C19MAPT
SCHEMBL16025801 0.71 ELANE (0.44) MAPK1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL31522409 0.71 ACSS2 (0.45) MAPK1KDM4EALDH1A1HPGDRAB9A
SCHEMBL9986928 0.71 KDM4E (0.43) KDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1656079-A Pyrazole compounds and pharmaceutical compositions containing the same EISAI CO LTD (JP) 2005-08-17 CN disclosed