SCHEMBL27623948

SCHEMBL27623948

O=C(c1ccc(-c2ccccn2)o1)c1ccc(-c2ccccn2)o1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.50
FAAH O00519 4/20 0.47
CES1 P23141 3/20 0.47
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
CCR1 P32246 1/20 0.45
CCR5 P51681 1/20 0.45
CCR8 P51685 1/20 0.45
METAP1 P53582 1/20 0.45
BLM P54132 1/20 0.45
HIF1A Q16665 1/20 0.45
DOHH Q9BU89 1/20 0.45
P4HTM Q9NXG6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3589894 0.88 ALDH1A1 (0.54) ALOX5FAAHCES1KDM4E
SCHEMBL3055621 0.86 ALOX5 (0.48) ALOX5FAAHCES1KDM4ELMNA
SCHEMBL27568458 0.86 ALOX5 (0.55) ALOX5FAAHCES1KDM4ELMNA
SCHEMBL3076222 0.80 KDM4E (0.62) ALOX5KDM4ELMNACYP1A2POLB
SCHEMBL3589756 0.79 LMNA (0.51) ALOX5KDM4ELMNA
Hexane SCHEMBL8813158 0.79 FAAH (0.49) FAAHCES1
SCHEMBL30387679 0.72 KDM4E (0.50) ALOX5KDM4ELMNACYP1A2POLB
SCHEMBL5224048 0.72 NPC1 (0.64) ALOX5KDM4ELMNACYP1A2POLB
SCHEMBL624039 0.71 PIK3CA (0.55) ALOX5KDM4ELMNACYP1A2POLB
SCHEMBL14999169 0.71 PDE4A (0.46) ALOX5KDM4ELMNACYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed