SCHEMBL27626733

SCHEMBL27626733

Cc1ccc(C(C=O)CBr)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 3/20 0.35
CASR P41180 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPA1 O75762 1/20 0.32
LMNA P02545 1/20 0.32
CHRM1 P11229 1/20 0.32
SLC6A2 P23975 1/20 0.32
ADRA1A P35348 1/20 0.32
HTR2B P41595 1/20 0.32
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CACNA1G O43497 1/20 0.32
CACNA2D1 P54289 1/20 0.32
CACNA1B Q00975 1/20 0.32
CACNB1 Q02641 1/20 0.32
CACNA1C Q13936 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27607823 0.83 ESR2 (0.41) SRCCHRM1ADRA1AHTR2B
SCHEMBL27549906 0.78 ESR1 (0.41) MEN1KMT2ALMNACHRM1SLC6A2
SCHEMBL28017568 0.77 HTR1A (0.40) SLC6A2TDP1ALDH1A1
SCHEMBL3413433 0.76 TDP1 (0.35) SRCCASRMEN1KMT2ATRPA1
SCHEMBL27546845 0.73 CYP2A6 (0.38) MEN1KMT2ALMNATDP1SMN1; SMN2
SCHEMBL27766137 0.73 TRPA1 (0.41) SRCCASRTRPA1LMNACHRM1
SCHEMBL27624254 0.72 MEN1 (0.31) MEN1KMT2AALDH1A1
SCHEMBL27624261 0.72 CYP3A4 (0.36) LMNAHTR2BTP53TDP1SMN1; SMN2
SCHEMBL27605513 0.71 ACP3 (0.40) TP53TDP1HTTALDH1A1
SCHEMBL27626730 0.71 SMN1; SMN2 (0.40) SRCMEN1KMT2ATRPA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101611005-A Be used as the acetophenones of the replacement of PDE4 inhibitor LEO PHARMA AS (DK) 2009-12-23 CN disclosed
CN-100381429-C Thiazole derivatives HOFFMANN LA ROCHE (CH) 2008-04-16 CN disclosed
CN-1946703-A Substituted thiazole and pyrimidine derivatives as melanocortin receptor modulators TRANSTECH PHARMA INC (US) 2007-04-11 CN disclosed
CN-1675188-A Thiazole derivatives HOFFMANN LA ROCHE (CH) 2005-09-28 CN disclosed