SCHEMBL27627481

SCHEMBL27627481

Cc1cccc(CC(C=O)c2ccc3nnn(C)c3c2)n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.37
CYP11B1 P15538 1/20 0.37
KEAP1 Q14145 6/20 0.36
SLC9A1 P19634 1/20 0.36
NOTUM Q6P988 1/20 0.35
NSD2 O96028 1/20 0.34
PDE8B O95263 1/20 0.34
BRD4 O60885 2/20 0.32
NFE2L2 Q16236 2/20 0.31
HCAR3 P49019 1/20 0.31
TGFBR1 P36897 1/20 0.31
BRD2 P25440 1/20 0.31
BRD3 Q15059 1/20 0.31
BRDT Q58F21 1/20 0.31
GRM4 Q14833 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27627479 0.84 CYP19A1 (0.38) CYP19A1CYP11B1KEAP1SLC9A1NOTUM
SCHEMBL6224234 0.80 CYP19A1 (0.38) CYP19A1CYP11B1KEAP1SLC9A1NOTUM
SCHEMBL27565161 0.80 TGFBR1 (0.41) BRD4TGFBR1
SCHEMBL27608277 0.74 SLC9A1 (0.41) KEAP1SLC9A1NOTUMNSD2TGFBR1
SCHEMBL4065212 0.73 HCAR3 (0.42) KEAP1SLC9A1NOTUMNSD2BRD4
SCHEMBL27584907 0.73 GRM5 (0.39) TGFBR1
SCHEMBL15341829 0.68 CYP19A1 (0.50) CYP19A1CYP11B1KEAP1SLC9A1NOTUM
SCHEMBL9523659 0.66 CYP19A1 (0.50) CYP19A1CYP11B1KEAP1SLC9A1NSD2
SCHEMBL4029836 0.64 TGFBR1 (0.38) KEAP1SLC9A1TGFBR1
SCHEMBL4032039 0.64 FAAH (0.38) KEAP1SLC9A1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1681805-A Novel imidazole compounds as transforming growth factor (TGF) inhibitors PFIZER PROD INC (US) 2005-10-12 CN disclosed