SCHEMBL27633455

SCHEMBL27633455

[CH2]c1cnn(-c2ccc(-c3ccccc3)nc2)c1-c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.39
PTGS1 P23219 2/20 0.38
PTGS2 P35354 2/20 0.38
CHRNB2 P17787 2/20 0.37
CHRNA7 P36544 2/20 0.37
CHRNA4 P43681 2/20 0.37
NPC1 O15118 3/20 0.35
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
PKM P14618 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
NFKB2 Q00653 1/20 0.33
KMT2A Q03164 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HIF1A Q16665 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28757409 0.93 S1PR1 (0.40) S1PR1PTGS1PTGS2NPC1MEN1
SCHEMBL5907261 0.85 PTGS2 (0.45) S1PR1PTGS1PTGS2NPC1RAB9A
SCHEMBL27653952 0.82 MAP4K1 (0.43) S1PR1PTGS1PTGS2CHRNB2CHRNA7
SCHEMBL5907288 0.82 PTGS2 (0.36) S1PR1PTGS1PTGS2CHRNB2CHRNA7
SCHEMBL5907422 0.77 CHRNB2 (0.39) S1PR1CHRNB2CHRNA7CHRNA4NPC1
SCHEMBL5907410 0.77 PDCD1 (0.38) S1PR1PTGS1PTGS2CHRNB2CHRNA7
SCHEMBL5907378 0.77 ALDH1A1 (0.42) PTGS2CHRNB2CHRNA7CHRNA4L3MBTL1
SCHEMBL5907360 0.75 ALDH1A1 (0.60) NPC1RAB9AMEN1NFKB1NFKB2
SCHEMBL5907291 0.75 MAP4K1 (0.41) CHRNB2CHRNA7CHRNA4L3MBTL1MAPT
SCHEMBL5907388 0.75 SSTR5 (0.37) CHRNB2CHRNA7CHRNA4L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1768051-A Substituted pyrazoles MERCK PATENT GMBH (DE) 2006-05-03 CN disclosed