SCHEMBL28757409

SCHEMBL28757409

[CH2]c1cnn(-c2ccc(-c3ccc(F)cc3)nc2)c1-c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.40
NR3C1 P04150 5/20 0.37
PGR P06401 2/20 0.37
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
NPC1 O15118 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
DHODH Q02127 1/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GRM4 Q14833 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
CYP17A1 P05093 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27633455 0.93 S1PR1 (0.39) S1PR1NPSR1L3MBTL1NPC1DHODH
SCHEMBL5907261 0.81 PTGS2 (0.45) S1PR1NR3C1PGRLMNANPSR1
SCHEMBL7262216 0.76 HTR2C (0.40) L3MBTL1MAPT
SCHEMBL5741014 0.76 CYP2A13 (0.43) LMNAL3MBTL1NPC1MAPTALOX5AP
SCHEMBL5907297 0.76 FABP3 (0.38) S1PR1NR3C1LMNANPSR1NPC1
SCHEMBL27653952 0.75 MAP4K1 (0.43) S1PR1L3MBTL1NPC1MAPTALOX5AP
SCHEMBL5907288 0.75 PTGS2 (0.36) S1PR1NPC1DHODHMEN1KMT2A
SCHEMBL5907378 0.70 ALDH1A1 (0.42) L3MBTL1PTGS2
SCHEMBL5907410 0.70 PDCD1 (0.38) S1PR1NPC1ALOX5APFEN1PTGS1
SCHEMBL5907422 0.70 CHRNB2 (0.39) S1PR1NPSR1L3MBTL1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1768051-A Substituted pyrazoles MERCK PATENT GMBH (DE) 2006-05-03 CN disclosed