SCHEMBL27633486

SCHEMBL27633486

CS(=O)(=O)c1nc(-c2ccccc2)c(C(=O)c2[nH]c(S(C)(=O)=O)nc2-c2ccccc2)[nH]1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.65
HPGD P15428 1/20 0.65
PTGS2 P35354 7/20 0.57
PTGS1 P23219 6/20 0.57
PIN1 Q13526 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
NPBWR1 P48145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5759689 0.91 ALDH1A1 (0.69) ALDH1A1HPGDPTGS2PTGS1PIN1
SCHEMBL6495602 0.82 ALDH1A1 (0.55) ALDH1A1HPGDPTGS2PTGS1SMN1; SMN2
SCHEMBL14692202 0.78 PTGS2 (0.63) ALDH1A1HPGDPTGS2PTGS1SMN1; SMN2
SCHEMBL27653921 0.77 HPGD (0.58) ALDH1A1HPGDPIN1SMN1; SMN2
SCHEMBL20376677 0.76 ALDH1A1 (0.50) ALDH1A1HPGDPTGS2PTGS1SMN1; SMN2
SCHEMBL27653935 0.75 CYP1A2 (0.42) ALDH1A1HPGDPIN1SMN1; SMN2
SCHEMBL27653989 0.70 TAAR1 (0.62) ALDH1A1HPGDPIN1SMN1; SMN2
SCHEMBL27633484 0.68 KDM4E (0.37) ALDH1A1HPGDPIN1
SCHEMBL5762947 0.67 KDM4E (0.62) ALDH1A1HPGDPIN1SMN1; SMN2
SCHEMBL4752688 0.66 HPGD (0.41) ALDH1A1HPGDPTGS2PTGS1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100427472-C Aryl-heteroaromatic compounds, compositions containing them and their use AVENTIS PHARMA SA (FR) 2008-10-22 CN claimed
CN-1829697-A Aryl-heteroaromatic products, compositions containing same and use thereof AVENTIS PHARMA SA (FR) 2006-09-06 CN claimed
CN-100427472-C Aryl-heteroaromatic compounds, compositions containing them and their use AVENTIS PHARMA SA (FR) 2008-10-22 CN disclosed
CN-1829697-A Aryl-heteroaromatic products, compositions containing same and use thereof AVENTIS PHARMA SA (FR) 2006-09-06 CN disclosed