SCHEMBL27633484

SCHEMBL27633484

O=C(c1[nH]c(C[SH](=O)=O)nc1-c1ccccc1)c1[nH]c(C[SH](=O)=O)nc1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.37
TAAR1 Q96RJ0 2/20 0.36
CYP1A2 P05177 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
CYP2C19 P33261 1/20 0.36
PIN1 Q13526 1/20 0.36
PTGES O14684 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 3/20 0.35
RAB9A P51151 2/20 0.35
KMT2A Q03164 3/20 0.34
NR4A2 P43354 2/20 0.34
MEN1 O00255 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
NR4A1 P22736 1/20 0.34
NR4A3 Q92570 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27653935 0.74 CYP1A2 (0.42) KDM4ETAAR1CYP1A2MAPK1CASP1
SCHEMBL11050965 0.72 ADORA3 (0.51) KDM4ETAAR1PIN1PTGESLMNA
SCHEMBL27653921 0.72 HPGD (0.58) KDM4ECYP1A2MAPK1CASP1CYP2C19
SCHEMBL4802255 0.72 SMN1; SMN2 (0.49) KDM4ECYP1A2MAPK1CASP1CYP2C19
SCHEMBL11054392 0.72 SMN1; SMN2 (0.49) KDM4EPIN1RAB9AKMT2AMEN1
SCHEMBL27653989 0.69 TAAR1 (0.62) KDM4ETAAR1CYP1A2MAPK1CASP1
SCHEMBL27633486 0.68 ALDH1A1 (0.65) PIN1ALDH1A1HPGD
SCHEMBL27488851 0.66 LMNA (0.43) KDM4ECYP1A2MAPK1CYP2C19LMNA
SCHEMBL2337944 0.65 PIN1 (0.45) PIN1RAB9AKMT2ANR4A2MEN1
SCHEMBL6503776 0.64 PIN1 (0.50) KDM4ECYP1A2MAPK1CASP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100427472-C Aryl-heteroaromatic compounds, compositions containing them and their use AVENTIS PHARMA SA (FR) 2008-10-22 CN claimed
CN-1829697-A Aryl-heteroaromatic products, compositions containing same and use thereof AVENTIS PHARMA SA (FR) 2006-09-06 CN claimed
CN-100427472-C Aryl-heteroaromatic compounds, compositions containing them and their use AVENTIS PHARMA SA (FR) 2008-10-22 CN disclosed
CN-1829697-A Aryl-heteroaromatic products, compositions containing same and use thereof AVENTIS PHARMA SA (FR) 2006-09-06 CN disclosed