SCHEMBL2763375

SCHEMBL2763375

CN(C1CCN(C(=O)OC(C)(C)C)CC1)S(=O)(=O)C1CC1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.48
HPGD P15428 1/20 0.47
GPR119 Q8TDV5 13/20 0.46
USP2 O75604 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
EPHX1 P07099 1/20 0.45
MGLL Q99685 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL672670 0.92 USP30 (0.49) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL15170539 0.92 USP30 (0.49) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL24392051 0.85 GPR119 (0.53) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL1182635 0.85 GPR119 (0.51) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL31691545 0.84 DDB1 (0.44) HPGDGPR119USP2SMN1; SMN2
SCHEMBL56423 0.84 HPGD (0.50) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL29181777 0.83 HPGD (0.47) RECQLHPGDGPR119EPHX1
SCHEMBL4711418 0.80 HPGD (0.55) RECQLHPGDGPR119USP2SMN1; SMN2
SCHEMBL18418307 0.80 MGLL (0.71) RECQLUSP2SMN1; SMN2MGLL
SCHEMBL24393339 0.80 GPR119 (0.47) RECQLHPGDGPR119EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2176237-A1 PHTHALAZINONE DERIVATIVES AS INHIBITORS OF PARP-1 AstraZeneca AB (SE) 2010-04-21 EP disclosed
US-20090023727-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 2009-01-22 US disclosed
US-20090023727-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 2009-01-22 US disclosed
US-20090023727-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 2009-01-22 US disclosed
WO-2009004356-A1 PHTHALAZINONE DERIVATIVES AS INHIBITORS OF PARP-1 ASTRAZENECA AB (SE) 2009-01-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023727-A1 PHTHALAZINONE DERIVATIVES NR0B2, NR0B1, NR2E1 RECQL 1687/4885HPGD 1239/4885GPR119 893/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.