SCHEMBL27635358

SCHEMBL27635358

O=CC1(F)CCCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.44
KDM1A O60341 3/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
SIGMAR1 Q99720 6/20 0.39
TSHR P16473 2/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
DRD2 P14416 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2B P41595 1/20 0.38
MTOR P42345 1/20 0.38
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6495897 0.75 KDM1A (0.51) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL4862191 0.75 MEN1 (0.53) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL6667048 0.75 KDM1A (0.50) AKR1B1KDM1AMEN1KMT2ASIGMAR1
Hydrochloric Acid SCHEMBL4427642 0.74 KDM1A (0.50) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL2091146 0.72 KDM1A (0.45) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL21479899 0.71 MEN1 (0.42) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL18192167 0.69 SIGMAR1 (0.60) MEN1KMT2ASIGMAR1TSHRTP53
SCHEMBL31052615 0.69 SIGMAR1 (0.60) MEN1KMT2ASIGMAR1TSHRTP53
SCHEMBL19577941 0.68 KDM1A (0.47) AKR1B1KDM1AMEN1KMT2ASIGMAR1
SCHEMBL8745709 0.68 HDAC9 (0.46) AKR1B1KDM1AMEN1KMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102245562-B Process for the synthesis of amino-methyltetralin derivatives HOFFMANN LA ROCHE 2014-08-13 CN disclosed
CN-101119965-B Tetralin and indane derivatives and uses thereof HOFFMANN LA ROCHE 2012-09-26 CN disclosed
CN-102245562-A Process for the synthesis of amino-methyltetralin derivatives HOFFMANN LA ROCHE 2011-11-16 CN disclosed
CN-101472884-A 1 2 3 4-tetralin and indane derivatives and uses thereof HOFFMANN LA ROCHE (CH) 2009-07-01 CN disclosed
CN-100422181-C [1,8] naphthyridin-2-ones and related compounds for the treatment of schizophrenia WARNER LAMBERT CO (US) 2008-10-01 CN disclosed
CN-101119965-A Tetralin and indane derivatives and uses thereof ROCHE PALO ALTO LLC (CH) 2008-02-06 CN disclosed
CN-1839134-A [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia WARNER LAMBERT CO (US) 2006-09-27 CN disclosed