SCHEMBL27636552

SCHEMBL27636552

Nc1nn(Br)c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
POLB P06746 1/20 0.36
LIMK1 P53667 1/20 0.36
GAA P10253 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 2/20 0.35
GLA P06280 1/20 0.35
RECQL P46063 1/20 0.35
TTK P33981 1/20 0.35
GPR3 P46089 1/20 0.34
PDPK1 O15530 1/20 0.34
CYP3A4 P08684 1/20 0.34
PDGFRA P16234 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL628648 0.76 KDM4E (0.42) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL31298641 0.74 GPR3 (0.34) KDM4EALDH1A1HSD17B10POLBMAPT
SCHEMBL10371646 0.74 KDM4E (0.41) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL13030846 0.74 KDM4E (0.41) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL823488 0.74 GSK3B (0.45) KDM4EALDH1A1HSD17B10HPGDLIMK1
SCHEMBL10831975 0.71 MAPT (0.47) KDM4EALDH1A1HSD17B10NPC1RAB9A
SCHEMBL10103719 0.69 MPO (0.42) ALDH1A1HSD17B10HPGDKMT2ASMN1; SMN2
SCHEMBL4420492 0.69 PRKD3 (0.43) KDM4EALDH1A1HSD17B10HPGDLIMK1
SCHEMBL14216404 0.69 SLC9A1 (0.43) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL28823953 0.69 ALDH1A1 (0.38) KDM4EALDH1A1HSD17B10HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103080093-A Indazole compounds and their uses DANA FARBER CANCER INST INC 2013-05-01 CN disclosed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed