SCHEMBL27637672

SCHEMBL27637672

CN(C)CC(=C(C=O)c1cccc(F)c1)c1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 1/20 0.41
KMT2A Q03164 2/20 0.40
CYP2C9 P11712 6/20 0.37
CYP3A4 P08684 5/20 0.37
CYP2D6 P10635 5/20 0.37
CYP1A2 P05177 4/20 0.37
CYP2C19 P33261 4/20 0.37
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
HIF1A Q16665 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
GSK3B P49841 1/20 0.35
PARP1 P09874 1/20 0.35
GRK2 P25098 1/20 0.34
GRK3 P35626 1/20 0.34
USP2 O75604 2/20 0.34
TBXAS1 P24557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27337618 0.84 LTA4H (0.45) GRM1KMT2ACYP1A2CYP2C19ALDH1A1
SCHEMBL27523731 0.84 LTA4H (0.45) GRM1KMT2ACYP1A2CYP2C19ALDH1A1
SCHEMBL28777062 0.84 CES2 (0.35) KMT2ACYP3A4ALDH1A1CES2CES1
SCHEMBL27608101 0.80 KCNQ3 (0.45) KMT2ACYP2C9CYP2D6CYP1A2CYP2C19
SCHEMBL13504693 0.78 GRM1 (0.43) GRM1KMT2ACYP2C9CYP3A4CYP2D6
SCHEMBL27555390 0.76 BCL2L1 (0.37) GRM1KMT2ACYP1A2CYP2C19ALDH1A1
SCHEMBL27593338 0.73 TP53 (0.42) KMT2ACYP2C9CYP3A4CYP2D6CYP1A2
SCHEMBL27516306 0.71 POLB (0.41) ALDH1A1MAOAMAOBPARP1HPGD
SCHEMBL27555371 0.71 POLB (0.41) ALDH1A1MAOAMAOBPARP1HPGD
SCHEMBL27919066 0.70 RAB9A (0.37) KMT2AALDH1A1TSHRUSP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100519552-C Pyrazole compounds UBE INDUSTRIES (JP) 2009-07-29 CN disclosed
CN-1684953-A Pyrazole compounds UBE INDUSTRIES (JP) 2005-10-19 CN disclosed