SCHEMBL13504693

SCHEMBL13504693

CN(C)C(=C(C=O)c1ccncc1)c1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 1/20 0.43
KMT2A Q03164 1/20 0.42
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
CYP2C9 P11712 4/20 0.39
CYP1A2 P05177 4/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2D6 P10635 3/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP2C19 P33261 4/20 0.38
PARP1 P09874 1/20 0.37
USP2 O75604 1/20 0.37
GSK3B P49841 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PLA2G7 Q13093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5788690 0.83 LTA4H (0.49) GRM1KMT2ACYP1A2ALDH1A1CYP2C19
SCHEMBL27637672 0.78 GRM1 (0.41) GRM1KMT2ACES2CES1CYP2C9
SCHEMBL5353608 0.70 CES2 (0.50) GRM1KMT2ACES2CES1CYP2C9
SCHEMBL5353609 0.70 CES2 (0.50) GRM1KMT2ACES2CES1CYP2C9
SCHEMBL3068393 0.70 CES2 (0.74) GRM1KMT2ACES2CES1CYP2C9
SCHEMBL10920829 0.70 HTT (0.47) KMT2ACYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL10919795 0.70 HTT (0.47) KMT2ACYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL2044451 0.69 ALDH1A1 (0.43) KMT2ATSHRALDH1A1GSK3B
SCHEMBL11159920 0.66 POLB (0.67) KMT2ACES2CES1CYP1A2CYP3A4
SCHEMBL11159914 0.66 POLB (0.67) KMT2ACES2CES1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553096-B1 PYRAZOLE COMPOUNDS UBE INDUSTRIES (JP) 2012-10-31 EP disclosed