SCHEMBL27646258

SCHEMBL27646258

CC(=O)Oc1ccc(Cl)c(O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.56
LMNA P02545 3/20 0.48
KDM4E B2RXH2 5/20 0.47
FLT3 P36888 1/20 0.46
ACHE P22303 2/20 0.46
CA2 P00918 2/20 0.45
GLA P06280 2/20 0.45
GAA P10253 2/20 0.45
MAPT P10636 4/20 0.44
POLB P06746 2/20 0.44
PKM P14618 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 1/20 0.43
TTR P02766 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377507 0.85 CYP3A4 (0.52) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL473532 0.84 LMNA (0.52) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL50809 0.82 CYP3A4 (0.62) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL28890049 0.81 MEN1 (0.53) CYP3A4KDM4ECA2PKMTDP1
SCHEMBL29001439 0.81 KDM4E (0.61) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL1846855 0.81 MCL1 (0.57) CYP3A4LMNAKDM4EACHEGLA
SCHEMBL3331532 0.79 CHRNA3 (0.49) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL27593853 0.79 LMNA (0.47) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL12316409 0.79 LMNA (0.47) CYP3A4LMNAKDM4EFLT3ACHE
SCHEMBL21921357 0.78 CYP3A4 (0.58) CYP3A4LMNAKDM4EACHEGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101326161-B Novel compounds ASTRAZENECA AB 2013-04-17 CN disclosed
CN-100469769-C Benzyl-pyridazinons as reverse transcriptase inhibitors ROCHE PALO ALTO LLC (CH) 2009-03-18 CN disclosed
CN-101374804-A Substituted diphenylethers, -amines, -sulfides and -methanes for the treatment of respiratory disease ASTRAZENECA AB (SE) 2009-02-25 CN disclosed
CN-101326161-A Novel compounds ASTRAZENECA AB (SE) 2008-12-17 CN disclosed
CN-100406007-C Asthma and allergic inflammation modulators AMGEN INC (US) 2008-07-30 CN disclosed
CN-1764649-A Benzyl-pyridazinones as reverse transcriptase inhibitors ROCHE PALO ALTO LLC (CH) 2006-04-26 CN disclosed