Piperazine

Piperazine

SCHEMBL27656709

C1CNCCN1.COS(=O)(=O)O

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
NFKB1 P19838 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRA6 Q16445 1/20 0.40
HIF1A Q16665 1/20 0.35
MAPT P10636 1/20 0.35
PDE4A P27815 1/20 0.35
KDR P35968 1/20 0.35
CA2 P00918 2/20 0.35
USP2 O75604 1/20 0.35
CA1 P00915 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
CXCR4 P61073 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperazine SCHEMBL27727092 0.97 TSHR (0.39) TSHRLMNACYP3A4GABRA1GABRG2
Pyrrolidine SCHEMBL3839669 0.89 ALDH1A1 (0.40) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL6046913 0.89 TSHR (0.32) TSHRLMNACYP3A4GABRA1GABRG2
Piperidine SCHEMBL30496139 0.87 ALDH1A1 (0.45) TSHRLMNACYP3A4GABRA1GABRG2
Piperidine SCHEMBL28253499 0.87 ALDH1A1 (0.45) TSHRLMNACYP3A4GABRA1GABRG2
Morpholine SCHEMBL9984285 0.83 MEN1 (0.48) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL3733571 0.81 HTR2C (0.33) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL27308161 0.80 TSHR (0.50) TSHRCYP3A4CA2USP2CA1
SCHEMBL27346657 0.80 TSHR (0.50) TSHRCYP3A4CA2USP2CA1
SCHEMBL5991 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929895-A Hypoxanthine and xanthine concentration analysis enzymatic compositions as the purine metabolism object for diagnosing tumor 高普生物有限公司 2018-12-04 CN claimed
CN-108179173-A A kind of mycobacterium tuberculosis susceptibility detection color developing agent and its susceptibility detection method 武汉轻工大学 2018-06-19 CN claimed
CN-107484643-A A kind of peony seeds breed breeding culture medium 安徽省雷氏农业科技有限公司 2017-12-19 CN claimed
EP-4736255-A2 SPIROBISINDANE COPOLYMERS AND METHODS OF MAKING Sepion Technologies, Inc. (US) 2026-05-06 EP disclosed
WO-2025006736-A9 SPIROBISINDANE COPOLYMERS AND METHODS OF MAKING SEPION TECHNOLOGIES, INC. (US) 2025-04-17 WO disclosed
WO-2025006736-A2 SPIROBISINDANE COPOLYMERS AND METHODS OF MAKING SEPION TECHNOLOGIES, INC. (US) 2025-01-02 WO disclosed
CN-106676123-B A kind of screening technique of glucose dehydrogenase mutant 厦门大学 2019-10-22 CN disclosed
CN-106323875-B Sample uses maximized system and method 西拉诺斯知识产权有限责任公司 2019-07-09 CN disclosed
CN-109897840-A Polyphosphoric acid dependent form glucokinase enzyme variants and its application 中国科学院天津工业生物技术研究所 2019-06-18 CN disclosed
CN-109689648-A 2-substituted benzothiazolyl-3-substituted phenyl-5-substituted sulfonated phenyl-2H-tetrazolium salt, reagent for measuring concentration of biological component containing the salt, and method for measuring concentration of biological component using the salt 泰尔茂株式会社 2019-04-26 CN disclosed
CN-104619851-B Method for producing methacrylic acid ester 三菱化学株式会社 2019-03-19 CN disclosed
CN-106255692-A Imidazo [4,5-c ] quinolin-2-one compounds and their use in treating cancer 阿斯利康(瑞典)有限公司 2016-12-21 CN disclosed
CN-103649754-B Assay method 杜邦营养生物科学有限公司 2016-11-02 CN disclosed
CN-103842518-B For the redox reagent compositions of electrochemica biological sensor and comprise the biosensor of described compositions 爱-森斯株式会社 2016-10-12 CN disclosed
CN-104427991-A Peptides derived from HIV GP41 for the treatment of T cell mediated pathologies YEDA RES & DEV 2015-03-18 CN disclosed
CN-103477197-A System and method for maximizing sample usage THERANOS INC 2013-12-25 CN disclosed
CN-101108809-B 1- (alkylaminoalkyl-pyrrolidine-/piperidinyl) -2, 2-diphenylacetamide derivatives as muscarinic receptor antagonists THERAVANCE INC 2010-07-14 CN disclosed
CN-100406435-C 1- (alkylaminoalkyl-pyrrolidine-/piperidinyl) -2, 2-diphenylacetamide derivatives as muscarinic receptor antagonists THERAVANCE INC (US) 2008-07-30 CN disclosed
CN-101108809-A 1- (alkylaminoalkyl-pyrrolidine-/piperidinyl) -2, 2-diphenylacetamide derivatives as muscarinic receptor antagonists THERAVANCE INC (US) 2008-01-23 CN disclosed
CN-1805927-A 1- (alkylaminoalkyl-pyrrolidine-/piperidinyl) -2, 2-diphenylacetamide derivatives as muscarinic receptor antagonists THERAVANCE INC (US) 2006-07-19 CN disclosed