SCHEMBL27664664

SCHEMBL27664664

COc1ccc(N(C(=O)c2ccccc2Cl)c2nc(C(=O)N3CCSCC3)c(C)s2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
HTR2C P28335 1/20 0.36
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
SPTLC2 O15270 5/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE4B Q07343 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27664670 0.91 HTR2C (0.47) NPC1RAB9AHTR2CTSHRMAPT
SCHEMBL5032532 0.91 NPC1 (0.37) NPC1RAB9ALMNATSHRMAPT
SCHEMBL27664668 0.86 POLB (0.43) NPC1RAB9ALMNATSHRSPTLC2
SCHEMBL27664673 0.84 NPC1 (0.41) NPC1RAB9ACES2CES1HTR2C
SCHEMBL5035881 0.84 KMT2A (0.39) NPC1RAB9ALMNAMAPTKMT2A
SCHEMBL5032530 0.82 HTR2C (0.43) NPC1RAB9AHTR2CTP53MAPT
SCHEMBL5035249 0.79 LMNA (0.38) NPC1RAB9ALMNAMAPTKMT2A
SCHEMBL5034690 0.79 CNR1 (0.40) NPC1RAB9ALMNASPTLC2KMT2A
SCHEMBL27664739 0.77 HTR2C (0.52) NPC1RAB9AHTR2CLMNATP53
SCHEMBL5032649 0.77 ALDH1A1 (0.48) NPC1RAB9ALMNATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN claimed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN claimed
CN-100509808-C Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2009-07-08 CN disclosed
CN-1890236-A Novel thiazole derivates HOFFMANN LA ROCHE (CH) 2007-01-03 CN disclosed