SCHEMBL27669147

SCHEMBL27669147

CCCCC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 3/20 0.71
CTSK P43235 7/20 0.60
CTSS P25774 4/20 0.60
CTSB P07858 2/20 0.60
CTSL P07711 1/20 0.60
ATM Q13315 1/20 0.53
AKT1 P31749 1/20 0.53
KLK5 Q9Y337 1/20 0.51
REN P00797 1/20 0.51
PPARG P37231 1/20 0.50
PPARA Q07869 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323726 0.90 ACE (0.71) ACECTSKCTSSCTSBCTSL
SCHEMBL1791039 0.87 ACE (0.78) ACECTSKCTSSCTSBCTSL
SCHEMBL7326335 0.87 ACE (0.78) ACECTSKCTSSCTSBCTSL
SCHEMBL2603668 0.87 ACE (0.70) ACECTSKCTSSCTSBCTSL
SCHEMBL9262578 0.86 ACE (0.65) ACECTSKCTSSCTSBCTSL
SCHEMBL1790253 0.84 ACE (0.70) ACECTSKCTSSCTSBCTSL
SCHEMBL6516027 0.84 ACE (0.70) ACECTSKCTSSCTSBCTSL
SCHEMBL17688687 0.84 ACE (0.70) ACECTSKCTSSCTSBCTSL
SCHEMBL10536264 0.84 ACE (0.70) ACECTSKCTSSCTSBCTSL
SCHEMBL8271187 0.84 CTSK (0.59) ACECTSKCTSSCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100537523-C Phenylamide and pyridylamide beta-secretase inhibitors for the treatment of alzheimer's disease MERCK & CO INC (US) 2009-09-09 CN disclosed
CN-1898199-A Phenylamide and pyridylamide beta-secretase inhibitors for the treatment of alzheimer's disease MERCK & CO INC (US) 2007-01-17 CN disclosed