SCHEMBL27671995

SCHEMBL27671995

CC(C)CNC(CCC(F)c1ccccc1)C(=O)NCC#N

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 14/20 0.53
CTSL P07711 12/20 0.53
CTSK P43235 10/20 0.53
CTSB P07858 9/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3873085 0.74 CTSS (0.51) CTSSCTSLCTSKCTSB
SCHEMBL17365596 0.71 CTSS (0.56) CTSSCTSLCTSKCTSB
SCHEMBL17365565 0.71 CTSS (0.56) CTSSCTSLCTSKCTSB
SCHEMBL2155836 0.69 CTSL (1.00) CTSSCTSLCTSKCTSB
SCHEMBL12681974 0.68 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL12681870 0.68 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL4718865 0.67 CTSK (0.78) CTSSCTSLCTSKCTSB
SCHEMBL7330779 0.67 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL6447090 0.67 CTSK (0.58) CTSSCTSLCTSKCTSB
SCHEMBL5526073 0.66 CTSK (0.62) CTSSCTSLCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1898219-A Novel keto-oxadiazole derivatives as cathepsin inhibitors AVENTIS PHARMA INC (US) 2007-01-17 CN claimed
CN-100543017-C Keto-oxadiazole derivatives as cathepsin inhibitors AVENTIS PHARMA INC (US) 2009-09-23 CN disclosed
CN-1898219-A Novel keto-oxadiazole derivatives as cathepsin inhibitors AVENTIS PHARMA INC (US) 2007-01-17 CN disclosed