SCHEMBL2767332

SCHEMBL2767332

Cc1cccc(Cl)c1NC(=S)Nc1noc2cc(F)ccc12

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 6/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
CHRNA7 P36544 5/20 0.41
TP53 P04637 3/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LCK P06239 1/20 0.37
RAB9A P51151 1/20 0.36
HTR3A P46098 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772968 0.80 SMN1; SMN2 (0.41) LMNASMN1; SMN2ALDH1A1CHRNA7TP53
SCHEMBL2767333 0.75 TP53 (0.42) SMN1; SMN2CHRNA7TP53RAB9AHTR3A
SCHEMBL2787077 0.75 CHRNA7 (0.43) GAACHRNA7LCK
SCHEMBL2769741 0.73 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1MAPTTP53CACNA1B
SCHEMBL2768955 0.72 MAOB (0.52) GAALMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL2767526 0.72 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1MAPTCHRNA7TP53
SCHEMBL8496098 0.70 RAB9A (0.71) GAALMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL2769004 0.68 PPIA (0.49) GAASMN1; SMN2ALDH1A1MAPTTP53
SCHEMBL2767338 0.68 KMT2A (0.52) GAALMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL2768640 0.67 MAPT (0.50) GAASMN1; SMN2ALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881967-B1 SUBSTITUTED BENZO(D)ISOXAZOL-3-YL AMINE COMPOUNDS AS ANALGESICS GRUENENTHAL GMBH (DE) 2010-04-28 EP claimed
US-20080176915-A1 Substituted Benzo[d]isoxazol-3-yl Amine Compounds as Analgesics GRUENENTHAL GMBH (DE) 2008-07-24 US claimed
US-7696238-B2 Substituted benzo[d]isoxazol-3-yl amine compounds as analgesics GRUENENTHAL GMBH (DE) 2010-04-13 US disclosed
US-20080176915-A1 Substituted Benzo[d]isoxazol-3-yl Amine Compounds as Analgesics GRUENENTHAL GMBH (DE) 2008-07-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176915-A1 Substituted Benzo[d]isoxazol-3-yl Amine Compounds as Analgesics KCNQ1, KCNQ2, KCNQ3 GAA 3898/4885LMNA 1716/4885SMN1; SMN2 1349/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.