SCHEMBL27675146

SCHEMBL27675146

O=C(O)c1cn(C(=O)Nc2ccc(Cl)nc2)c2ccccc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 6/20 0.47
KCNQ2 O43526 6/20 0.47
CHRM1 P11229 3/20 0.45
LMNA P02545 1/20 0.44
KCNE1 P15382 4/20 0.41
KCNQ1 P51787 4/20 0.41
MAOB P27338 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.39
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28766931 0.85 CHRM1 (0.52) CHRM1LMNAMAOBKDM4E
SCHEMBL27693500 0.84 CHRM1 (0.41) CHRM1LMNAMAOBKDM4E
SCHEMBL27675094 0.84 TRPV1 (0.45) CHRM1LMNAKDM4E
SCHEMBL27693487 0.83 LMNA (0.51) CHRM1LMNAMAOBKDM4EALDH1A1
SCHEMBL27675384 0.82 CHRM1 (0.49) CHRM1LMNAMAOBKDM4EALDH1A1
SCHEMBL27675247 0.82 NPC1 (0.47) CHRM1LMNAKDM4EALDH1A1
SCHEMBL27675121 0.80 CHRM1 (0.47) CHRM1LMNAKDM4E
SCHEMBL27693452 0.80 CHRM1 (0.49) CHRM1LMNAMAOBKDM4E
SCHEMBL27675102 0.80 LMNA (0.44) LMNAALDH1A1
SCHEMBL27693534 0.80 MAOB (0.50) CHRM1LMNAMAOBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed