SCHEMBL27675203

SCHEMBL27675203

CCCCc1ccc(C=O)cc1[N+](=O)[O-]

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 2/20 0.57
ALDH5A1 P51649 1/20 0.53
ABAT P80404 1/20 0.53
VCAM1 P19320 1/20 0.53
ALDH1A1 P00352 10/20 0.47
TDP1 Q9NUW8 2/20 0.47
MAPT P10636 7/20 0.46
ALDH1A3 P47895 1/20 0.46
LMNA P02545 4/20 0.43
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
XDH P47989 1/20 0.41
PDK1 Q15118 1/20 0.38
TTR P02766 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27841940 0.89 ALDH3A1 (0.52) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL2924523 0.87 ALDH3A1 (0.62) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL17922571 0.82 ALDH1A1 (0.58) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL30353219 0.82 ALDH1A1 (0.58) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL27780985 0.81 ALDH5A1 (0.56) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL5080802 0.80 TYR (0.43) ALDH3A1ALDH1A1TDP1MAPTALDH1A3
SCHEMBL4575571 0.79 ALDH5A1 (0.62) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL6355056 0.79 ALDH5A1 (0.57) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL8759780 0.79 ALDH5A1 (0.57) ALDH3A1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL8887647 0.79 ALDH1A1 (0.68) ALDH1A1TDP1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-103641765-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2014-03-19 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-102652128-A 4-Oxo-1H-quinoline-3-carboxamides as modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-08-29 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed