SCHEMBL27675233

SCHEMBL27675233

CN(C)c1cccc(NC(=O)n2cc(C(=O)O)c(=O)c3ccccc32)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CREBBP Q92793 3/20 0.47
EP300 Q09472 1/20 0.47
MAOB P27338 3/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
ALOX15 P16050 1/20 0.44
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
HIF1A Q16665 1/20 0.43
LMNA P02545 1/20 0.41
HTR6 P50406 1/20 0.40
CHRM1 P11229 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KCNK3 O14649 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675196 0.85 CREBBP (0.52) MEN1KMT2ACREBBPEP300MAOB
SCHEMBL27693487 0.85 LMNA (0.51) MEN1KMT2ACREBBPEP300MAOB
SCHEMBL27693516 0.84 CREBBP (0.61) MEN1KMT2ACREBBPEP300MAOB
SCHEMBL27693567 0.84 CREBBP (0.47) CREBBPEP300MAOBALDH1A1LMNA
SCHEMBL27675227 0.83 CFTR (0.48) CREBBPEP300MAOBALDH1A1LMNA
SCHEMBL27693586 0.83 MAOB (0.60) MEN1KMT2ACREBBPEP300MAOB
SCHEMBL27693520 0.83 CASP3 (0.52) MEN1KMT2ACREBBPEP300ALDH1A1
SCHEMBL27675135 0.82 CREBBP (0.54) MEN1KMT2ACREBBPEP300MAOB
SCHEMBL27675183 0.82 CREBBP (0.46) CREBBPEP300MAOBALDH1A1LMNA
SCHEMBL27693473 0.81 LMNA (0.50) CREBBPEP300MAOBLMNACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed