SCHEMBL27680698

SCHEMBL27680698

O=C(C(Cn1ccnc1)c1ccc(Br)cn1)C(Cn1ccnc1)c1ccc(Br)cn1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 1/20 0.47
CYP3A4 P08684 1/20 0.43
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PKM P14618 1/20 0.40
NOS1 P29475 1/20 0.39
FDPS P14324 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27956563 0.81 HMOX1 (0.62) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL27680700 0.80 HMOX1 (0.45) HMOX1CYP3A4CYP19A1CYP11B1CYP11B2
SCHEMBL27956576 0.80 MEN1 (0.45) FDPS
SCHEMBL27680695 0.74 ALPG (0.40)
SCHEMBL27660667 0.74 ALDH1A1 (0.43) KDM4EFDPS
SCHEMBL27680813 0.73 SMN1; SMN2 (0.44)
SCHEMBL27924984 0.72 CYP1A2 (0.38) CYP3A4KDM4E
SCHEMBL27961723 0.72 ALDH1A1 (0.42) KDM4EFDPS
SCHEMBL4554609 0.71 CYP19A1 (0.50) CYP19A1CYP11B1CYP11B2KDM4E
SCHEMBL27680699 0.71 RAB9A (0.36) MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679454-A Antimicrobial heterocyclic compounds for treatment of bacterial infections MICURX PHARMACEUTICALS INC 2010-03-24 CN disclosed
CN-1989137-A 3- '4- {6-substituted alkanoyl) pyridin-3-yl} -3-phenyl! -5- (1h-1, 2, 3-triazol-1-ylmethyl) -1, 3-oxazolidin-2-ones as antibacterial agents ASTRAZENECA AB (SE) 2007-06-27 CN disclosed