SCHEMBL27685281

SCHEMBL27685281

CC(C)NC(=O)N1CCN(Cc2ccc(F)cc2)C(=O)C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.62
DPP4 P27487 6/20 0.52
MCHR1 Q99705 1/20 0.49
CSNK1D P48730 1/20 0.46
CSNK1E P49674 1/20 0.46
RAB9A P51151 1/20 0.45
HTT P42858 1/20 0.44
HDAC1 Q13547 1/20 0.44
CYP3A4 P08684 1/20 0.43
MAPK1 P28482 1/20 0.43
FAAH O00519 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41
PRKAB1 Q9Y478 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2894836 0.86 DPP4 (0.52) TP53DPP4MCHR1RAB9AHTT
SCHEMBL3911313 0.82 DPP4 (0.55) TP53DPP4MCHR1RAB9AHTT
SCHEMBL27616276 0.80 DPP4 (0.56) TP53DPP4MCHR1RAB9AHTT
SCHEMBL4238855 0.78 DPP4 (0.46) TP53DPP4MCHR1RAB9AHTT
SCHEMBL15858005 0.76 ALDH1A1 (0.53) TP53DPP4MCHR1RAB9AHTT
SCHEMBL4158417 0.76 DPP4 (0.49) TP53DPP4MCHR1RAB9AHTT
SCHEMBL3906693 0.75 DPP4 (0.56) TP53DPP4MCHR1RAB9AHTT
SCHEMBL17897294 0.75 RAB9A (0.49) TP53DPP4MCHR1RAB9AHTT
SCHEMBL2899646 0.73 PKM (0.39) TP53CSNK1DCSNK1EHDAC1CYP3A4
SCHEMBL11640756 0.72 CACNA1G (0.46) DPP4HTTHDAC1CYP3A4FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1929737-A HIV integrase inhibitors MERCK & CO INC (US) 2007-03-14 CN disclosed