SCHEMBL27686159

SCHEMBL27686159

NC(=O)c1c(CC(O)O)c2ncc(Cc3ccc(F)cc3)cc2n(Cc2ccc(C[SH](=O)=O)cc2)c1=O

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.34
GRM2 Q14416 3/20 0.31
P2RX3 P56373 3/20 0.30
TNIK Q9UKE5 1/20 0.30
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686146 0.93 CNR2 (0.33) CNR2GRM2
SCHEMBL27666974 0.91 CNR2 (0.33) CNR2GRM2P2RX3TNIKCNR1
SCHEMBL28765661 0.90 GRM2 (0.36) CNR2GRM2
SCHEMBL27686112 0.87 CYP1A2 (0.33) CNR2CNR1
SCHEMBL27667115 0.86 OPRM1 (0.35) CNR2
SCHEMBL27686188 0.86 GRIN1 (0.40) GRM2
SCHEMBL27667073 0.84
SCHEMBL27686115 0.84 DPP4 (0.34) CNR2GRM2
SCHEMBL27686353 0.84 GRIN1 (0.38) GRM2
SCHEMBL27667153 0.83 TRPC5 (0.38) CNR2GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed