SCHEMBL27686353

SCHEMBL27686353

NC(=O)c1c(CC(O)O)c2ncc(Cc3ccc(F)cc3)cc2n(Cc2ccccn2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.38
GRIN2B Q13224 4/20 0.38
HTT P42858 1/20 0.38
S1PR3 Q99500 4/20 0.36
GRM2 Q14416 2/20 0.36
TP53 P04637 1/20 0.36
FEN1 P39748 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRA5 P31644 1/20 0.35
OPRM1 P35372 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.33
GFER P55789 1/20 0.33
PLA2G2A P14555 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686312 0.93 GRIN1 (0.37) GRIN1GRIN2BHTTS1PR3GRM2
SCHEMBL28765661 0.87 GRM2 (0.36) GRIN1GRIN2BGRM2FEN1KDM4E
SCHEMBL27686188 0.87 GRIN1 (0.40) GRIN1GRIN2BGRM2FEN1GABRA1
SCHEMBL27686094 0.86 S1PR3 (0.39) GRIN1GRIN2BHTTS1PR3GRM2
SCHEMBL27667139 0.85 GRIN1 (0.37) GRIN1GRIN2BHTTS1PR3GRM2
SCHEMBL27686159 0.84 CNR2 (0.34) GRM2
SCHEMBL27686115 0.84 DPP4 (0.34) GRIN2BHTTGRM2KDM4EALDH1A1
SCHEMBL27667153 0.83 TRPC5 (0.38) GRM2
SCHEMBL27686289 0.82 LMNA (0.33) GRIN1GRIN2BGRM2LMNA
SCHEMBL27685962 0.81 MEN1 (0.37) GRIN2BGRM2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed