SCHEMBL27688784

SCHEMBL27688784

CCC1(C(=O)OCc2ccccc2N)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
USP30 Q70CQ3 1/20 0.40
TSHR P16473 2/20 0.39
SMARCA2 P51531 1/20 0.39
SMARCA4 P51532 1/20 0.39
PBRM1 Q86U86 1/20 0.39
ALOX15 P16050 1/20 0.39
ATM Q13315 1/20 0.39
MEN1 O00255 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
GPR119 Q8TDV5 2/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3182059 0.85 RAB9A (0.49) MEN1RAB9AKMT2A
SCHEMBL22014536 0.84 TACR1 (0.48) TACR1OPRD1OPRK1TSHRALOX15
SCHEMBL25295847 0.84 P2RX3 (0.42) TACR1OPRD1OPRK1TSHRALOX15
SCHEMBL22770414 0.82 POLB (0.46) OPRD1OPRK1MEN1RAB9AKMT2A
SCHEMBL25301984 0.82 POLB (0.43) OPRD1OPRK1RAB9AGPR119PKM
SCHEMBL28528706 0.78 P2RX7 (0.43) TACR1GPR119PKM
SCHEMBL28986539 0.78 USP2 (0.45) TACR1OPRD1OPRK1PKM
SCHEMBL963907 0.78 USP2 (0.47) TSHRMEN1KMT2APKM
SCHEMBL20608062 0.77 USP30 (0.41) TACR1OPRD1OPRK1USP30TSHR
SCHEMBL28974232 0.77 NAMPT (0.54) OPRD1OPRK1MEN1KMT2AGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101072771-B Cgrp receptor antagonists MERCK & CO INC 2010-09-29 CN disclosed
CN-101072771-A Cgrp receptor antagonists MERCK & CO INC (US) 2007-11-14 CN disclosed