SCHEMBL2769600

SCHEMBL2769600

O=C(O)[C@@H](O)Cc1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 1/20 0.56
CPA1 P15085 1/20 0.53
PPARG P37231 2/20 0.49
PPARA Q07869 2/20 0.49
ALDH1A1 P00352 1/20 0.46
TRPA1 O75762 1/20 0.46
FFAR1 O14842 1/20 0.44
ACE P12821 1/20 0.44
KMT2A Q03164 1/20 0.43
CTBP2 P56545 1/20 0.43
MME P08473 1/20 0.42
CA2 P00918 1/20 0.42
TPH1 P17752 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8953439 1.00 KDM6B (0.56) KDM6BCPA1PPARGPPARAALDH1A1
SCHEMBL1906641 1.00 KDM6B (0.56) KDM6BCPA1PPARGPPARAALDH1A1
SCHEMBL1906640 1.00 KDM6B (0.56) KDM6BCPA1PPARGPPARAALDH1A1
SCHEMBL18248073 0.94 KDM6B (0.51) KDM6BCPA1PPARGPPARAALDH1A1
SCHEMBL28815028 0.94 KDM6B (0.51) KDM6BCPA1PPARGPPARAALDH1A1
SCHEMBL10891346 0.89 KDM6B (0.67) KDM6BACEMME
SCHEMBL754625 0.83 LDHA (0.57) CPA1PPARGPPARAALDH1A1TRPA1
SCHEMBL1907744 0.82 EPHX1 (0.45) CPA1PPARGPPARATRPA1
SCHEMBL5807390 0.82 TRPA1 (0.48) KDM6BCPA1PPARGPPARATRPA1
SCHEMBL235131 0.81 KDM6B (0.63) KDM6BACEMMECA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883720-B2 Template-fixed beta-hairpin peptidomimetics with CXCR4 antagonizing activity POLYPHOR AG (CH) 2014-11-11 US disclosed
US-20110312879-A1 TEMPLATE-FIXED BETA-HAIRPIN PEPTIDOMIMETICS WITH CXCR4 ANTAGONIZING ACTIVITY POLYPHOR AG (CH) 2011-12-22 US disclosed
WO-2010060479-A1 TEMPLATE-FIXED BETA-HAIRPIN PEPTIDOMIMETICS WITH CXCR4 ANTAGONIZING ACTIVITY POLYPHOR AG (CH) 2010-06-03 WO disclosed
EP-1639119-B1 METHOD FOR THE MICROBIOLOGICAL ISOMERISATION OF ALPHA-HYDROXY CARBOXYLIC ACIDS BASF SE (DE) 2010-04-21 EP disclosed
EP-1639119-A1 METHOD FOR THE MICROBIOLOGICAL ISOMERISATION OF ALPHA-HYDROXY CARBOXYLIC ACIDS BASF AKTIENGESELLSCHAFT (DE) 2006-03-29 EP disclosed
WO-2004111257-A1 METHOD FOR THE MICROBIOLOGICAL ISOMERISATION OF ALPHA-HYDROXY CARBOXYLIC ACIDS BASF AKTIENGESELLSCHAFT (DE) 2004-12-23 WO disclosed
EP-1073672-A1 ANTIPICORNAVIRAL COMPOUNDS, THEIR PREPARATION AND USE AGOURON PHARMACEUTICALS, INC. (US) 2001-02-07 EP disclosed
WO-1999057135-A1 ANTIPICORNAVIRAL COMPOUNDS, THEIR PREPARATION AND USE AGOURON PHARMACEUTICALS, INC. (US) 1999-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110312879-A1 TEMPLATE-FIXED BETA-HAIRPIN PEPTIDOMIMETICS WITH CXCR4 ANTAGONIZING ACTIVITY CXCL12, CXCR4, CXCR1 KDM6B 4503/4885CPA1 340/4885PPARG 1778/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.