SCHEMBL27697649

SCHEMBL27697649

COC(=O)Cc1c[nH]c2cc(C)cc(C)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
NR4A2 P43354 2/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.40
NPC1 O15118 2/20 0.37
PDGFRB P09619 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37
FLT1 P17948 1/20 0.37
FGFR3 P22607 1/20 0.37
KDR P35968 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2673123 0.83 KDM4E (0.55) KDM4EMAPTPOLBGAANPSR1
SCHEMBL2847756 0.82 ICMT (0.51) KDM4EMAPTPOLBGAANPSR1
SCHEMBL9157807 0.80 KDM4E (0.46) KDM4EMAPTPOLBPDGFRBFGFR1
SCHEMBL14564356 0.77 NR4A2 (0.58) KDM4EMAPTNR4A2PKMNPC1
SCHEMBL3267595 0.74 HTR2C (0.44) KDM4EMAPTPOLBNPC1GPR17
SCHEMBL21255987 0.73 MTNR1A (0.59) KDM4EMAPTNR4A2POLBPKM
SCHEMBL6064603 0.72 MTNR1A (0.37) KDM4EMAPTPOLBPKMMTNR1A
SCHEMBL27531827 0.72 GPR17 (0.42) KDM4EMAPTNR4A2PKMMTNR1A
SCHEMBL20551235 0.71 KMT2A (0.51) KDM4EMAPTPOLBPKMCASP1
SCHEMBL9756250 0.71 NR4A2 (0.43) KDM4EMAPTNR4A2POLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101018781-A Bicyclic N-anilide spirolactam CGRP receptor antagonists MERCK & CO INC (US) 2007-08-15 CN disclosed