SCHEMBL27701412

SCHEMBL27701412

O=C1C[C](c2ccccc2)CCN1C(F)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
CFTR P13569 1/20 0.32
GOPC Q9HD26 1/20 0.32
ADRA1B P35368 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MCOLN3 Q8TDD5 1/20 0.31
PARL Q9H300 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758698 0.79 CHRM2 (0.49) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL28041982 0.66 CYP2D6 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL6580284 0.65 CYP3A4 (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL25356698 0.65 HSD11B1 (0.49) CYP3A4CYP2C19KMT2AALDH1A1MAPT
SCHEMBL25356702 0.65 HSD11B1 (0.49) CYP3A4CYP2C19KMT2AALDH1A1MAPT
SCHEMBL28945789 0.63 CHRM2 (0.33) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL1825079 0.62 DRD1 (0.52) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL915178 0.61 DPP4 (0.47) RAB9ALMNA
SCHEMBL11038239 0.61 CHRM2 (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8549438 0.60 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101014574-A HIV integrase inhibitors MERCK & CO INC (US) 2007-08-08 CN disclosed