SCHEMBL27705689

SCHEMBL27705689

CC(C)C(CCC(=O)ON)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.35
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
CYP2D6 P10635 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27696266 1.00 NOS1 (0.35) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL27437737 0.83 NOS1 (0.36) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL763872 0.81 GABRP (0.41) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL16350129 0.81 GABRP (0.41) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL27586297 0.78 MEN1 (0.36) NOS1NOS3NOS2
SCHEMBL9644345 0.77 NOS1 (0.32) NOS1NOS3NOS2
SCHEMBL27535928 0.75 CA1 (0.36) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL19919876 0.75 CPB2 (0.41) NOS1NOS3NOS2CA1CA2
SCHEMBL27899114 0.75 CYP2D6 (0.36) NOS1NOS3NOS2CYP2D6CA1
SCHEMBL28795933 0.74 CTSK (0.44) CA1CA2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101035770-B 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA NV 2011-02-23 CN disclosed
CN-101035770-A Novel 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2007-09-12 CN disclosed
CN-101035771-A 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE) JANSSEN PHARMACEUTICA NV (BE) 2007-09-12 CN disclosed