SCHEMBL27720191

SCHEMBL27720191

CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cccc(Cl)c3)cc2)ccc1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 3/20 0.55
RAF1 P04049 1/20 0.54
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
BRAF P15056 2/20 0.52
HDAC1 Q13547 2/20 0.52
KDR P35968 2/20 0.52
TEK Q02763 1/20 0.52
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
MAPT P10636 6/20 0.51
RAB9A P51151 5/20 0.51
LMNA P02545 4/20 0.51
HTT P42858 4/20 0.51
NPC1 O15118 4/20 0.51
ALDH1A1 P00352 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
PLK4 O00444 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27740983 0.90 CDK8 (0.56) CDK8RAF1BRAFHDAC1KDR
SCHEMBL27720100 0.90 BRAF (0.63) CDK8RAF1CA9BRAFHDAC1
SCHEMBL27720157 0.89 MAPT (0.64) CDK8RAF1CA2CA9BRAF
SCHEMBL27720144 0.88 TP53 (0.62) CDK8RAF1BRAFHDAC1MEN1
SCHEMBL27720155 0.86 BRAF (0.64) CDK8RAF1CA12CA1CA2
SCHEMBL27720117 0.85 BRAF (0.61) RAF1BRAFHDAC1MEN1KMT2A
SCHEMBL27720129 0.85 MEN1 (0.66) CDK8RAF1CA9BRAFHDAC1
SCHEMBL27720178 0.83 RAB9A (0.60) CDK8RAF1CA12CA1CA2
SCHEMBL27720106 0.83 RAF1 (0.51) CDK8RAF1CA9BRAFHDAC1
SCHEMBL16628069 0.81 KDR (0.73) CDK8RAF1CA9BRAFKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101298427-B Diaryl urea compound and use thereof GUANGZHOU INST BIOMED & HEALTH 2012-03-21 CN disclosed
CN-101298427-A Diaryl urea compound and use thereof GUANGZHOU INST BIOMED & HEALTH (CN) 2008-11-05 CN disclosed