SCHEMBL27720252

SCHEMBL27720252

NCc1ccc(Br)c(C[O])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA12 O43570 2/20 0.38
CA4 P22748 2/20 0.38
CA6 P23280 2/20 0.38
CA5A P35218 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
CA5B Q9Y2D0 2/20 0.38
MAPT P10636 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
LOXL2 Q9Y4K0 3/20 0.34
HDAC3 O15379 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
CA3 P07451 1/20 0.34
CSNK2A1 P68400 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27839471 0.83 CA1 (0.33) CA1CA2CA12CA4CA6
SCHEMBL849381 0.83 CSNK2A1 (0.45) CA1CA2CA12CA4CA6
SCHEMBL27778402 0.79 ABAT (0.38) CA1CA2CA12CA4CA6
SCHEMBL27271778 0.75 CSNK2A1 (0.45) GAAPKMLOXL2CSNK2A1CSNK2A2
SCHEMBL29875339 0.75 HRH3 (0.43) CA1CA2CA12CA4CA6
SCHEMBL28958238 0.75 HRH3 (0.43) CA1CA2CA12CA4CA6
SCHEMBL28783294 0.75 LOXL2 (0.39) CA1CA2CA12CA4CA6
SCHEMBL1047304 0.73 HSP90AA1 (0.46) CA1CA2CA12CA9MAPT
SCHEMBL25383151 0.71 IDO1 (0.31)
SCHEMBL13443566 0.71 HRH3 (0.40) CA1CA2CA12CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101171230-A Heterocyclic-substituted alkanamides useful as renin inhibitors SPEEDEL EXPERIMENTA AG (CH) 2008-04-30 CN disclosed