SCHEMBL27720302

SCHEMBL27720302

N#Cc1cccc(-c2c[c]cnc2)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.50
CLK4 Q9HAZ1 1/20 0.49
GABRG2 P18507 7/20 0.48
GABRB3 P28472 7/20 0.48
GABRA5 P31644 7/20 0.48
GABRA3 P34903 7/20 0.48
GABRA1 P14867 1/20 0.48
CHRNB2 P17787 1/20 0.46
CHRNA5 P30532 1/20 0.46
CHRNA4 P43681 1/20 0.46
CYP17A1 P05093 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
NEK1 Q96PY6 1/20 0.43
NOTUM Q6P988 1/20 0.43
MAOB P27338 1/20 0.43
GRM5 P41594 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2750910 0.82 CYP11B2 (0.36) IDO1CLK4CHRNB2CHRNA5CHRNA4
SCHEMBL18890284 0.79 IDO1 (0.56) IDO1CLK4GABRG2GABRB3GABRA5
SCHEMBL5323457 0.79 CYP11B2 (0.55) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL2154026 0.78 CLK4 (0.65) IDO1CLK4GABRG2GABRB3GABRA5
SCHEMBL13537172 0.77 CYP11B2 (0.71) IDO1CLK4GABRG2GABRB3GABRA5
SCHEMBL29809001 0.77 CYP11B2 (0.71) IDO1CLK4GABRG2GABRB3GABRA5
SCHEMBL3721866 0.76 HSD17B1 (0.50) CYP17A1CYP11B1CYP11B2
SCHEMBL1201514 0.76 CYP11B2 (0.45) IDO1GABRG2GABRB3GABRA5GABRA3
SCHEMBL28800800 0.76 IDO1 (0.45) IDO1NOTUMMAOB
SCHEMBL27787243 0.75 CLK4 (0.63) IDO1CLK4GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103068797-B Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application SANOFI SA 2015-03-11 CN claimed
CN-103068797-B Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application SANOFI SA 2015-03-11 CN disclosed
CN-103068797-A Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application SANOFI SA 2013-04-24 CN disclosed
CN-101146817-B Novel compounds derived from 5-thioxylose and therapeutic use thereof FOURNIER LAB SA 2011-08-17 CN disclosed
CN-101146817-A Novel compounds derived from 5-thioxylose and therapeutic use thereof FOURNIER LAB SA (FR) 2008-03-19 CN disclosed