SCHEMBL27722334

SCHEMBL27722334

CCc1ccc(C)n2c(NCC(=O)NO)c(Cc3ccccc3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.36
HDAC8 Q9BY41 4/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
PKM P14618 1/20 0.35
HDAC1 Q13547 4/20 0.34
GRK2 P25098 1/20 0.34
PLA2G1B P04054 1/20 0.34
HDAC3 O15379 2/20 0.33
MMP9 P14780 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27722333 0.85 PKM (0.33) HDAC6HDAC8PKMHDAC1HDAC3
SCHEMBL27701649 0.83 HDAC1 (0.37) HDAC6HDAC8PKMHDAC1HDAC3
SCHEMBL28768873 0.81 HDAC6 (0.38) HDAC6HDAC8MEN1KMT2APKM
SCHEMBL28772858 0.77 HDAC8 (0.37) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL27701698 0.76 HDAC8 (0.45) HDAC8MEN1KMT2APLA2G1BCYP3A4
SCHEMBL27701659 0.75 HDAC6 (0.37) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL27722270 0.73 HDAC6 (0.39) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL27722212 0.73 PLAU (0.39) HDAC6HDAC8MEN1KMT2AHDAC1
SCHEMBL27701823 0.73 HDAC6 (0.38) HDAC6HDAC8MEN1KMT2ARXFP1
SCHEMBL27701646 0.73 PLAU (0.39) HDAC6HDAC8MEN1KMT2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101163703-B Imidazo [1,2-A ] pyridine derivatives as Peptide Deformylase (PDF) inhibitors NOVARTIS AG 2010-12-15 CN disclosed
CN-101163703-A Imidazo [1, 2-A ] pyridine derivatives as Peptide Deformylase (PDF) inhibitors NOVARTIS AG (CH) 2008-04-16 CN disclosed