SCHEMBL27723296

SCHEMBL27723296

O=Cc1cn(S(=O)(=O)CC=Cc2cccnc2)c(-c2ccccc2F)c1I

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.40
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TBXAS1 P24557 1/20 0.32
CHRNB2 P17787 2/20 0.32
CHRNA4 P43681 2/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA7 P36544 1/20 0.32
MEN1 O00255 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27744007 0.91 NFE2L2 (0.42) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL27723412 0.89 NFE2L2 (0.40) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL28031577 0.85 NFE2L2 (0.42) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL27723249 0.81 NFE2L2 (0.38) NFE2L2CYP11B1CYP11B2ALDH1A1MAPT
SCHEMBL27744280 0.81 NFE2L2 (0.43) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL27723315 0.80 NFE2L2 (0.35) NFE2L2CYP11B1CYP11B2TBXAS1CHRNB2
SCHEMBL1278426 0.79 CHRNB2 (0.36) NFE2L2ALDH1A1HTTSMN1; SMN2CHRNB2
SCHEMBL27723313 0.77 NFE2L2 (0.40) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL27744003 0.77 DCTPP1 (0.38) NFE2L2CYP11B1CYP11B2ALDH1A1MAPT
SCHEMBL27743986 0.76 NFE2L2 (0.40) NFE2L2CYP11B1CYP11B2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101300229-B 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL 2011-10-05 CN disclosed
CN-101300229-A 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL (JP) 2008-11-05 CN disclosed