SCHEMBL27744003

SCHEMBL27744003

Cc1c(C=O)cn(S(=O)(=O)CC=Cc2cccnc2)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCTPP1 Q9H773 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP1B1 Q16678 1/20 0.36
TBXAS1 P24557 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27723249 0.88 NFE2L2 (0.38) DCTPP1ALDH1A1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL27744007 0.79 NFE2L2 (0.42) ALDH1A1SMN1; SMN2CYP11B1CYP11B2CHRNB2
SCHEMBL27723224 0.78 CYP11B1 (0.40) DCTPP1ALDH1A1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL27744024 0.78 TBXAS1 (0.38) DCTPP1ALDH1A1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL1156646 0.77 KDM4E (0.41) ALDH1A1SMN1; SMN2CYP11B1CYP11B2CYP2C9
SCHEMBL27744045 0.77 TSHR (0.30) PTGS2
SCHEMBL27723296 0.77 NFE2L2 (0.40) ALDH1A1SMN1; SMN2CYP11B1CYP11B2CHRNB2
SCHEMBL27723299 0.77 CHRNB2 (0.41) DCTPP1CYP11B1CYP11B2CHRNB2CHRNA4
SCHEMBL27723412 0.77 NFE2L2 (0.40) ALDH1A1SMN1; SMN2CYP11B1CYP11B2CHRNB2
SCHEMBL27723432 0.76 L3MBTL1 (0.38) ALDH1A1SMN1; SMN2CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101300229-B 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL 2011-10-05 CN disclosed
CN-101300229-A 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors TAKEDA PHARMACEUTICAL (JP) 2008-11-05 CN disclosed