SCHEMBL27726697

SCHEMBL27726697

CC(c1ccc2ccccc2c1)c1nc(N)nc(N)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.50
ADRA2A P08913 3/20 0.48
ADRA2B P18089 3/20 0.48
ADRA2C P18825 3/20 0.48
CYP1A2 P05177 2/20 0.42
HTR2A P28223 2/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
HTR6 P50406 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
AOC3 Q16853 2/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
ATM Q13315 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
ADORA2A P29274 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28806243 0.89 UGT2B7 (0.61) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL28567977 0.76 ADRA2A (0.51) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
Ammonia Solution, Strong SCHEMBL308383 0.75 SMN1; SMN2 (0.48) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL16746751 0.74 ADRA2A (0.47) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL3001927 0.74 UGT2B7 (0.61) UGT2B7ADRA2AADRA2BADRA2CCYP2D6
SCHEMBL918554 0.73 UGT2B7 (0.59) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL6836009 0.73 ESR1 (0.56) CYP1A2CYP2D6TSHRHIF1AADORA2A
SCHEMBL599956 0.72 UGT2B7 (0.71) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL30928206 0.72 UGT2B7 (0.71) UGT2B7ADRA2AADRA2BADRA2CCYP1A2
SCHEMBL9179436 0.72 UGT2B7 (0.71) UGT2B7ADRA2AADRA2BADRA2CCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103265495-A Multicyclic amino acid derivatives and methods of their use LEXICON GENETICS INC 2013-08-28 CN disclosed
CN-101351451-B Polycyclic amino acid derivatives and methods of use thereof LEXICON PHARMACEUTICALS INC 2013-02-20 CN disclosed
CN-101351451-A Polycyclic amino acid derivatives and methods of use thereof LEXICON GENETICS INC (US) 2009-01-21 CN disclosed