Acridine

Acridine

SCHEMBL2772852

O=[N+]([O-])O.O=[N+]([O-])O.c1ccc2nc3ccccc3cc2c1.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Acridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.65
HPGD P15428 3/20 0.65
MAPT P10636 3/20 0.65
GLA P06280 2/20 0.65
ACHE P22303 1/20 0.65
RAB9A P51151 3/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
HTR3A P46098 1/20 0.48
CYP3A4 P08684 1/20 0.45
NQO2 P16083 2/20 0.44
KDM4E B2RXH2 5/20 0.44
GAA P10253 3/20 0.44
STAT3 P40763 1/20 0.44
HTT P42858 1/20 0.43
ATM Q13315 1/20 0.43
IKBKB O14920 1/20 0.43
NPC1 O15118 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL27479824 1.00 ALDH1A1 (0.65) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL9106792 1.00 ALDH1A1 (0.65) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL31425247 1.00 ALDH1A1 (0.65) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL27479825 1.00 ALDH1A1 (0.65) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL28796207 0.98 ALDH1A1 (0.62) ALDH1A1HPGDMAPTGLAACHE
Acridine SCHEMBL28471035 0.87 ALDH1A1 (0.65) ALDH1A1HPGDMAPTGLAACHE
Nitric Acid SCHEMBL3888889 0.84 KMT2A (0.51) ALDH1A1HPGDMAPTGLAACHE
Anthracene SCHEMBL27489981 0.84 CYP3A4 (0.54) ALDH1A1HPGDGLARAB9AKMT2A
Acridine SCHEMBL27545385 0.83 RAB9A (0.63) ALDH1A1HPGDMAPTGLAACHE
Nitric Acid SCHEMBL3961222 0.81 KMT2A (0.49) ALDH1A1HPGDMAPTGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114391095-A Oxidase-based chemiluminescence assay of phagocytic leukocytes in whole blood and body fluids suitable for point-of-care (POC) measurement of Absolute Neutrophil Function (ANF) for point-of-care (POC) diagnostic tests 比纳瑞有限责任公司 2022-04-22 CN claimed
CN-108350466-B Methods and compositions for determining pH 芝加哥大学 2022-06-24 CN disclosed
CN-114391095-A Oxidase-based chemiluminescence assay of phagocytic leukocytes in whole blood and body fluids suitable for point-of-care (POC) measurement of Absolute Neutrophil Function (ANF) for point-of-care (POC) diagnostic tests 比纳瑞有限责任公司 2022-04-22 CN disclosed
CN-114391095-A Oxidase-based chemiluminescence assay of phagocytic leukocytes in whole blood and body fluids suitable for point-of-care (POC) measurement of Absolute Neutrophil Function (ANF) for point-of-care (POC) diagnostic tests 比纳瑞有限责任公司 2022-04-22 CN disclosed
EP-1549759-B1 BACTERIAL TEST METHOD BY GLYCATED INTRACELLULAR ENZYMES SIEMENS HEALTHCARE DIAGNOSTICS (US) 2010-04-28 EP disclosed
EP-1549759-A4 BACTERIAL TEST METHOD BY GLYCATED LABEL BINDING BAYER HEALTHCARE LLC (US) 2006-11-02 EP disclosed
US-20060141546-A1 Bacterial test method by glycated label binding SIEMENS HEALTHCARE DIAGNOSTICS INC. 2006-06-29 US disclosed
EP-1549759-A1 BACTERIAL TEST METHOD BY GLYCATED LABEL BINDING Bayer Healthcare LLC (US) 2005-07-06 EP disclosed
WO-2003106699-A1 BACTERIAL TEST METHOD BY GLYCATED LABEL BINDING BAYER HEALTHCARE LLC (US) 2003-12-24 WO disclosed
US-20030232401-A1 Bacterial test method by glycated label binding BAYER CORPORATION 2003-12-18 US disclosed
EP-0660876-A1 A PROCESS OF QUANTIFYING CELL NUMBER Packard Instrument Company, Inc. (US) 1995-07-05 EP disclosed
US-5306624-A Process of quantifying cell number PACKARD INSTRUMENT CO., INC. (US) 1994-04-26 US disclosed
WO-1994006932-A1 A PROCESS OF QUANTIFYING CELL NUMBER PACKARD INSTRUMENT COMPANY, INC. (US) 1994-03-31 WO disclosed