SCHEMBL27731900

SCHEMBL27731900

FC(F)(F)c1c[nH]c(-c2ccc(Cl)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PTGS1 P23219 3/20 0.41
PTGS2 P35354 3/20 0.41
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
ALPL P05186 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.39
HPGD P15428 1/20 0.38
FABP4 P15090 1/20 0.38
TYMP P19971 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11623789 0.91 HPGD (0.43) KDM4EALDH1A1HSD17B10HPGDTYMP
SCHEMBL26093883 0.84 KDM4E (0.44) KDM4EALDH1A1HSD17B10HPGDTYMP
SCHEMBL8797359 0.84 GFER (0.50) KDM4EHPGDTYMPNPC1RAB9A
SCHEMBL19625464 0.82 ALPL (0.43) KDM4EALDH1A1HSD17B10ALPLDCUN1D1
SCHEMBL16661274 0.82 KDM4E (0.45) KDM4EHPGDTYMPSMN1; SMN2NR1H2
SCHEMBL11626212 0.82 KIF11 (0.42) KDM4EALDH1A1HSD17B10HPGDNPC1
SCHEMBL3095172 0.82 HPGD (0.38) KDM4EPTGS2HPGDTYMPNPC1
SCHEMBL27731893 0.82 NPBWR1 (0.44) PTGS1PTGS2ALPLDCUN1D1HPGD
SCHEMBL649565 0.81 HPGD (0.56) KDM4EALDH1A1HSD17B10PTGS1KCNQ3
SCHEMBL29429388 0.81 NPC1 (0.44) KDM4EALDH1A1KCNQ3KCNQ2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101239981-B Pyrazolo and imidazo-pyrimidine derivatives HOFFMANN LA ROCHE 2011-01-19 CN disclosed
CN-100522964-C Pyrazolo and imidazo-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2009-08-05 CN disclosed
CN-101239981-A Pyrazolo and imidazo-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2008-08-13 CN disclosed