SCHEMBL27744690

SCHEMBL27744690

C=CC(N1CCN(c2ccc(C(F)(F)F)c(Cl)c2)CC1CC)S(=O)(=O)c1ccc2c(c1)C(C(=O)O)CC2

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.43
NR1H2 P55055 7/20 0.38
NR1H3 Q13133 7/20 0.38
HSD11B1 P28845 1/20 0.33
DPP4 P27487 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765780 0.93 NR1H2 (0.35) NOTUMNR1H2NR1H3HSD11B1
SCHEMBL27744699 0.87 NOTUM (0.44) NOTUMNR1H2NR1H3HSD11B1
SCHEMBL27765621 0.86 RORC (0.36) NOTUMNR1H2NR1H3
SCHEMBL27765640 0.85 NOTUM (0.42) NOTUMNR1H2NR1H3HSD11B1
SCHEMBL1471063 0.85 NOTUM (0.47) NOTUMNR1H2NR1H3HSD11B1
SCHEMBL28780732 0.82 SLC6A9 (0.35) HSD11B1
SCHEMBL27744574 0.82 F13A1 (0.39) NR1H2NR1H3DPP4
SCHEMBL27765691 0.79 NOTUM (0.36) NOTUMNR1H2NR1H3
SCHEMBL20309080 0.78 NOTUM (0.49) NOTUMNR1H2NR1H3DPP4
SCHEMBL1471118 0.78 HSD11B1 (0.41) NOTUMNR1H2NR1H3HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101421258-B Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYPSYS INC 2013-08-21 CN disclosed
CN-101421258-A Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYSPSYS INC (US) 2009-04-29 CN disclosed