SCHEMBL27744707

SCHEMBL27744707

C=CC(N1C(C)CN(c2ccc(C(F)(F)F)cc2)CC1C)S(=O)(=O)c1ccc2c(c1)C(C(=O)O)CC2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.36
SLC6A9 P48067 7/20 0.36
TRPA1 O75762 4/20 0.32
CACNA1B Q00975 1/20 0.32
HDAC1 Q13547 1/20 0.32
RORC P51449 2/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
KCNH2 Q12809 1/20 0.31
HTR6 P50406 1/20 0.31
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28780715 0.90 NOTUM (0.34) NOTUMRORC
SCHEMBL27765595 0.88 HSD11B1 (0.40) SLC6A9CA1CA2CA7CA9
SCHEMBL27765640 0.88 NOTUM (0.42) NOTUM
SCHEMBL27744659 0.86 SLC6A9 (0.41) NOTUMSLC6A9RORCCA1CA2
SCHEMBL1470752 0.83 NOTUM (0.41) NOTUMSLC6A9TRPA1HDAC1CHRM2
SCHEMBL1470754 0.83 NOTUM (0.41) NOTUMSLC6A9TRPA1HDAC1CHRM2
SCHEMBL20309069 0.83 NOTUM (0.41) NOTUMSLC6A9TRPA1HDAC1CHRM2
SCHEMBL27744761 0.79 F13A1 (0.34) SLC6A9RORCCA1CA2CA7
SCHEMBL27765644 0.78
SCHEMBL27744766 0.77 EGLN1 (0.34) RORCMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101421258-B Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYPSYS INC 2013-08-21 CN disclosed
CN-101421258-A Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYSPSYS INC (US) 2009-04-29 CN disclosed